产品描述: | SRPIN340 is an ATP-competitive serine-arginine-rich protein kinase (SRPK) inhibitor, with a Ki of 0.89 μM for SRPK1. |
靶点: |
Ki: 0.89 μM (SRPK1);VirusProtease;Serine/threoninkinase |
参考文献: |
1. Fukuhara T, et al. Utilization of host SR protein kinases and RNA-splicing machinery during viral replication. Proc Natl Acad Sci U S A. 2006 Jul 25;103(30):11329-33. 2. Siqueira RP, et al. Potential Antileukemia Effect and Structural Analyses of SRPK Inhibition by N-(2-(Piperidin-1-yl)-5-(Trifluoromethyl)Phenyl)Isonicotinamide (SRPIN340). PLoS One. 2015 Aug 5;10(8):e0134882. |
溶解性: |
DMSO : ≥ 42 mg/mL (120.22 mM) |
保存条件: |
2-8℃ |
配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
1 mM |
2.862 ml |
14.312 ml |
28.625 ml |
5 mM |
0.572 ml |
2.862 ml |
5.725 ml |
10 mM |
0.286 ml |
1.431 ml |
2.862 ml |
50 mM |
0.057 ml |
0.286 ml |
0.572 ml |
|
注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |