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产品描述： Tiapride hydrochloride is a selective and orally active D2 and D3 dopamine receptors antagonist with IC50 values of 110-320 nM and 180 nM, respectively. Tiapride hydrochloride shows anti-dyskinetic activity and anxiolytic activity. Tiapride hydrochloride is a neuroleptic agent |
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靶点：
D2 Receptor:110-320 nM (IC50);D3 Receptor:180 nM (IC50);DopamineReceptor |
参考文献：
1. Scatton B, et al. The preclinical pharmacologic profile of tiapride. Eur Psychiatry. 2001 Jan;16 Suppl 1:29s-34s. 2. Peters DH, et al. Tiapride. A review of its pharmacology and therapeutic potential in the management of alcohol dependence syndrome. Drugs. 1994 Jun;47(6):1010-32. |
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溶解性：
H2O : ≥ 200 mg/mL (548.11 mM) DMSO : 31.25 mg/mL (85.64 mM; Need ultrasonic) |
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保存条件：
-20℃ |
配置溶液浓度参考：
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1mg |
5mg |
10mg |
| 1 mM |
2.741 ml |
13.703 ml |
27.406 ml |
| 5 mM |
0.548 ml |
2.741 ml |
5.481 ml |
| 10 mM |
0.274 ml |
1.37 ml |
2.741 ml |
| 50 mM |
0.055 ml |
0.274 ml |
0.548 ml |
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| 注意： |
部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。 |
上海工商
北京