产品描述: | Skepinone-L is a selective p38 mitogen-activated protein kinase inhibitor. |
靶点: |
Autophagy;p38 MAPK;p38MAPK; Autophagy |
体内研究: |
In vivo, skepinone-L inhibits Gal/ LPS-induced TNF-α release by 77%. |
细胞实验: |
Concentrations: 1 nM - 10 μM, dissolved in DMSO |
参考文献: |
1.Koeberle SC, et al. Nat Chem Biol. 2011, 8(2), 141-143. 2.Borst O, et al. Cell Physiol Biochem. 2013, 31(6), 914-924. |
溶解性: |
H2O:<1 mg/mL Ethanol:79 mg/mL (185.7 mM) DMSO:79 mg/mL (185.7 mM) |
保存条件: |
-20℃ |
配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
1 mM |
2.351 ml |
11.753 ml |
23.506 ml |
5 mM |
0.47 ml |
2.351 ml |
4.701 ml |
10 mM |
0.235 ml |
1.175 ml |
2.351 ml |
50 mM |
0.047 ml |
0.235 ml |
0.47 ml |
|
注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |