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产品描述： CB-7921220 is an adenylate cyclase inhibitor. |
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靶点：
Adenylate Cyclase;AChR |
体外研究：
CB-7921220 shows a degree of isoform selectivity for adenylate cyclase (AC) 1, but cannot distinguish between AC1 and AC6. CB-7921220 has a more consistent predicted binding position in the two virtual docking screens, and has a binding conformation similar to ATP and P-site inhibitors, which may explain its lack of selectivity between AC1 and AC6 |
参考文献：
1. Brand CS, et al. Isoform selectivity of adenylyl cyclase inhibitors: characterization of known and novel compounds. J Pharmacol Exp Ther. 2013 Nov;347(2):265-75. |
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溶解性：
soluble in DMSO |
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保存条件：
-20℃ |
配置溶液浓度参考：
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1mg |
5mg |
10mg |
| 1 mM |
4.162 ml |
20.811 ml |
41.622 ml |
| 5 mM |
0.832 ml |
4.162 ml |
8.324 ml |
| 10 mM |
0.416 ml |
2.081 ml |
4.162 ml |
| 50 mM |
0.083 ml |
0.416 ml |
0.832 ml |
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| 注意： |
部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。 |
上海工商
危险品化学品经营许可证（不带存储）
营业执照(三证合一)
北京