产品描述: | Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer. |
靶点: |
mTOR; PI3K;PI3K; mTOR |
参考文献: |
1. Shao Z,et al. VS-5584, a Novel PI3K-mTOR Dual Inhibitor, Inhibits Melanoma Cell Growth In Vitro and In Vivo. PLoS One. 2015 Jul 23;10(7). 2. Kolev VN, et al. PI3K/mTOR dual inhibitor VS-5584 preferentially targets cancer stem cells. Cancer Res. 2015 Jan 15;75(2):446-55. |
溶解性: |
Soluble in DMSO |
保存条件: |
-20℃ |
配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
1 mM |
2.938 ml |
14.689 ml |
29.379 ml |
5 mM |
0.588 ml |
2.938 ml |
5.876 ml |
10 mM |
0.294 ml |
1.469 ml |
2.938 ml |
50 mM |
0.059 ml |
0.294 ml |
0.588 ml |
|
注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |