S83391 |
Cambinol |
源叶(MedMol) | 98% |
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- 产品描述: Cambinol is a SIRT1 and SIRT2 inhibitor with IC50 values of 56 μM and 59 μM, respectively. Cambinol is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibitor)
- 靶点: SIRT1:56 μM (IC50);SIRT2:59 μM (IC50);Apoptosis; Phospholipase; Sirtuin
- 体内研究:
Cambinol is well tolerated in mice (100 mg/kg) and inhibits growth of Burkitt lymphoma xenografts. No significant weight loss occurs in cambinol-treated animals relative to controls. Inhibitors of NAD-dependent deacetylases may constitute novel anticancer agents
- 参考文献:
1. Heltweg B, et al. Antitumor activity of a small-molecule inhibitor of human silent information regulator 2 enzymes. Cancer Res. 2006 Apr 15;66(8):4368-77. 2. Huarui Zhang, et al. Advances in the discovery of exosome inhibitors in cancer. J Enzyme Inhib Med Chem. 2020 Dec;35(1):1322-1330.
- 溶解性: DMSO : 50 mg/mL (138.72 mM; Need ultrasonic)
- 保存条件: RT
- 配置溶液浓度参考:
1mg 5mg 10mg 1 mM 2.774 ml 13.872 ml 27.745 ml 5 mM 0.555 ml 2.774 ml 5.549 ml 10 mM 0.277 ml 1.387 ml 2.774 ml 50 mM 0.055 ml 0.277 ml 0.555 ml
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本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为:
质量 (mg) = 浓度 (mM) x 体积 (mL) x 分子摩尔量 (g/mol)