S83445 |
Niraparib metabolite M1 |
源叶(MedMol) | 99% |
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- 产品描述: Niraparib metabolite M1 is a metabolite of niraparib, and the latter one acts as a novel poly(ADP-Ribose) polymerase (PARP) inhibitor.
- 靶点: Drug Metabolite;Others
- 体外研究:
Niraparib metabolite M1 has the validation in plasma and urine for the support of clinical studies such as the mass balance study and the absolute bioavailability study
- 参考文献:
1. van Andel L, et al. Liquid chromatography-tandem mass spectrometry assay for the quantification of niraparib and its metabolite M1 in human plasma and urine. J Chromatogr B Analyt Technol Biomed Life Sci. 2016 Nov 19;1040:14-21
- 溶解性: soluble in DMSO
- 保存条件: -20℃
- 配置溶液浓度参考:
1mg 5mg 10mg 1 mM 3.112 ml 15.558 ml 31.116 ml 5 mM 0.622 ml 3.112 ml 6.223 ml 10 mM 0.311 ml 1.556 ml 3.112 ml 50 mM 0.062 ml 0.311 ml 0.622 ml
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本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为:
质量 (mg) = 浓度 (mM) x 体积 (mL) x 分子摩尔量 (g/mol)