S83760 |
2-CL-IB-MECA |
源叶(MedMol) | 99% |
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- 产品描述: Namodenoson (CF-102) is a selective A3 adenosine receptor (A3AR) agonist (Ki=0.33 nM). Namodenoson displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively
- 靶点: Ki:0.33 nM (A3 adenosine receptor);AdenosineReceptor
- 体内研究:
Intravenous administration of 200 μg/kg Namodenoson (2-Cl-IB-MECA) resulted in a short-lasting hypotension, which was accompanied by a 50-100-fold increase in plasma histamine concentrations. Administration of a second dose of Namodenoson (2-Cl-IB-MECA) did not elicit any hemodynamic effects
- 参考文献:
1. Van Schaick EA et al. Hemodynamic effects and histamine release elicited by the selective adenosine A3 receptor agonist 2-Cl-IB-MECA in conscious rats. Eur J Pharmacol. 1996 Jul 25;308(3):311-4. 2. Jacobson KA et al. Adenosine A3 receptors: novel ligands and paradoxical effects. Trends Pharmacol Sci. 1998 May;19(5):184-91.
- 溶解性: DMSO : ≥ 31 mg/mL (56.91 mM)
- 保存条件: 2-8℃
- 配置溶液浓度参考:
1mg 5mg 10mg 1 mM 1.836 ml 9.179 ml 18.358 ml 5 mM 0.367 ml 1.836 ml 3.672 ml 10 mM 0.184 ml 0.918 ml 1.836 ml 50 mM 0.037 ml 0.184 ml 0.367 ml
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本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为:
质量 (mg) = 浓度 (mM) x 体积 (mL) x 分子摩尔量 (g/mol)